Targets：CFTR inhibitors medchemexpress products name :A-839977 GKT137831 Product alias :SYN-5005 Description: A-839977 is a potent, CNS penetrating P2X7 antagonist whixh blocks BzATP-evoked calcium influx at P2X7 receptors. (IC50 values are…
Targets：Calcium Channel inhibitors medchemexpress products name :VUF11207 TFA Salt PF-04447943 Product alias :SYN-5245 Description: High-potency ligand that induces recruitment of β-arrestin2 and subsequent internalization of CXCR7.cas no. : 1378524-41-4Api wt.…
Targets：BCRP inhibitors medchemexpress products name :VPC23019 PF-04418948 Product alias :SYN-5242 Description: Sphingosine-1-phosphate receptor antagonist.cas no. : 449173-19-7Api wt. : 372.40
Targets：ATP Synthase inhibitors medchemexpress products name :UNC2170 maleate GM6001 Product alias :SYN-5678 Description: A micromolar ligand for the Methyl-lysine Binding Protein 53BP1. .cas no. : 1648707-58-7 (free base)Api wt. :…
Targets：Membrane Transporter_Ion Channel inhibitors medchemexpress products name :RXFP1-Agonist GSK2606414 Product alias :SYN-5228 Description: The first potent and selective small-molecule agonist of human relaxin receptor 1 (RXFP1) A cell-permeable 2-acetamido-N-phenylbenzamide that…
Targets：Ribosomal S6 Kinase (RSK) inhibitors medchemexpress products name :Pyridostatin PLX8394 Product alias :SYN-5373 Description: Pyridostatin stabilizes G-quadruplexes targeting the proto-oncogene SRC and telomeric G-quadruplexes inducing DNA damage and cell-cycle arrest…
Targets：Raf inhibitors medchemexpress products name :Molindone Hydrochloride T-5224 Product alias :SYN-5562 Description: A D2DR inhibitor and a MAO inhibitor.cas no. : 15622-65-8Api wt. : 312.83
Targets：p38 MAPK inhibitors medchemexpress products name :ML 00253764 Hydrochloride EW-7197 Product alias :SYN-5200 Description: Non-peptide, melanocortin MC4 receptor antagonist (IC50 values are 0.32, 0.81 and 2.12 μM for MC4, MC3…
Targets：MNK inhibitors medchemexpress products name :JYL1421 EMD638683 Product alias :SYN-5011 Description: JYL1421 is a selective TRPV1 vanilloid receptor antagonist. Vanilloid receptors play a roll in sensory transduction for capsaicin (…
Targets：Mixed Lineage Kinase inhibitors medchemexpress products name :JTE-013 INCB3344 Product alias :SYN-5010 Description: Sphingosine-1-phosphate (S1P) receptor antagonist, highly selective for S1P2 (EDG-5). Inhibits S1P binding to human S1P2 receptors (IC50…